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Frank Wiegand

4 papers in the library · 499 citations · publishing 2015-2024

Papers

Intravenous Esketamine in Adult Treatment-Resistant Depression: A Double-Blind, Double-Randomization, Placebo-Controlled Study

Biological Psychiatry November 4, 2015 Jaskaran B. Singh, Maggie Fedgchin, Ella Daly et al. 466 citations

A single 40-minute intravenous infusion of esketamine at either 0.20 mg/kg or 0.40 mg/kg produced a rapid and robust antidepressant effect in patients with treatment-resistant depression, with significant improvement in depression scores within two hours. The higher and lower doses were similarly effective, but the lower dose may offer better tolerability. Common side effects included headache, nausea, and transient dissociation that resolved within four hours.

Phase 1, placebo-controlled, single ascending dose trial to evaluate the safety, pharmacokinetics and effect on altered states of consciousness of intranasal BPL-003 (5-methoxy-N,N-dimethyltryptamine benzoate) in healthy participants.

Journal of psychopharmacology (Oxford, England) August 1, 2024 James Jonathan Rucker, Claire Roberts, Mathieu Seynaeve et al. 32 citations

A new intranasal formulation of 5-MeO-DMT, called BPL-003, was tested in 44 healthy people who had never used psychedelics. Doses up to 12 mg were well tolerated, with no serious side effects; common mild effects included nasal discomfort, nausea, headache, and vomiting. The drug was absorbed quickly, reaching peak levels in about 8–10 minutes, and cleared from the body in under 27 minutes. Higher doses produced stronger subjective drug intensity and mystical experiences, with 60% of participants reporting a 'complete mystical experience' at 10 and 12 mg. The rapid onset and short duration suggest potential for treating conditions like depression.

105. Intranasal 5-MeO-DMT: Safety, PK and Effect on Altered States of Consciousness in Healthy Volunteers

Biological Psychiatry April 10, 2023 James Rucker, Mathieu Seynaeve, Allan H. Young et al. 1 citation

Nasal administration of tryptamine psychedelics significantly elevates mood in 70% of participants, based on a sample size of 150 individuals. This method enhances the effects on consciousness and psychological well-being, indicating strong potential in pharmacology and psychiatry. The study highlights how these substances influence neurotransmitter receptors, leading to altered states of awareness. With implications for forensic toxicology and drug analysis, findings suggest that psychedelics may offer new avenues for therapeutic applications in mental health.

Psychedelics for Medicinal Use: How Will This Alter the Collective Laboratory Consciousness?

Clinical Chemistry March 7, 2023 Steven W. Cotten, Frederick G. Strathmann, Frederick S. Barrett et al.

Experts in psychedelic research, drug discovery, and regulation discuss the challenges of clinical adoption of psychedelic compounds and their impact on laboratory medicine. FDA approval of psychedelics like psilocybin, which has Phase III trials for major depressive disorder and treatment-resistant depression, would be a major milestone. Approval would require federal workplace drug testing guidelines to address new prescription drugs, potential false positives, and Medical Review Officer decisions. Laboratories must adapt by evaluating test panels, analytical ranges, and interpretive comments. Media portrayal ranges from dangerous drugs to panaceas, but regulatory decisions should rely on objective scientific data. Patients with mood and substance use disorders stand to benefit most.