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Leandro J Bertoglio

Department of Pharmacology, Federal University of Santa Catarina, Florianopolis, Santa Catarina, Brazil.

3 papers in the library · 21 citations · publishing 2024-2026

Papers

Ayahuasca-enhanced extinction of fear behaviour: Role of infralimbic cortex 5-HT2A and 5-HT1A receptors.

British journal of pharmacology June 1, 2024 Isabel Werle, Laura M M Nascimento, Aymee L A Dos Santos et al. 21 citations

A single oral dose of ayahuasca containing 0.3 mg/kg of DMT increased within-session extinction of contextual freezing behavior in rats without affecting recall; two consecutive daily doses enhanced extinction recall. These effects occurred for both 1- and 21-day-old memories in males and females, independent of changes in anxiety or general exploratory activity. Blocking 5-HT2A receptors in the infralimbic cortex prevented within-session extinction, while blocking 5-HT1A receptors prevented between-session extinction. The findings highlight complementary mechanisms by which ayahuasca facilitates behavioral suppression of aversive memories, suggesting potential benefits for stress-related disorders.

Psychedelics and Mental Health in Endurance Athletes: A Cross-Sectional Study in Brazil.

Journal of psychoactive drugs March 20, 2026 Marina A M Portes, Leandro J Bertoglio

Endurance athletes face unique psychological and physical stressors, yet their knowledge and attitudes toward psychedelic therapies are largely unknown. A survey of 28 Brazilian endurance athletes (mean age 37) found that 64% reported a lack of mental health support in their athletic environments. Only 11% had prior psychedelic experience, while 79% were open to legal, supervised psychedelic therapies. However, 61% were unaware of evidence for psychedelics in treating mental health conditions, and 78% mistakenly believed psychedelics are addictive. Women more often reported pharmacological treatment for depression or anxiety. The findings highlight unmet mental health needs, knowledge gaps, and misconceptions, pointing to a need for targeted, evidence-based education.

Ayahuasca modulation of traumatic-like fear memories requires infralimbic cortex BDNF-dependent mechanisms in rats.

European neuropsychopharmacology : the journal of the European College of Neuropsychopharmacology February 1, 2026 Isabel Werle, Francisco S Guimarães, Rafael G Dos Santos et al.

Ayahuasca, a brew containing the psychedelic DMT, helps rodents overcome persistent and generalized fear memories by boosting brain-derived neurotrophic factor (BDNF) signaling in the infralimbic (IL) region of the medial prefrontal cortex. In rats exposed to stress or high-intensity fear conditioning, repeated ayahuasca (0.3 mg/kg DMT) enhanced extinction learning and its retention, and reduced fear generalization. These effects were blocked by infusing an anti-BDNF antibody or a TrkB receptor antagonist into the IL cortex. The reduction in fear generalization depended on BDNF in females but not males. The findings suggest psychedelics may aid in treating difficult-to-extinguish trauma memories, such as those in PTSD.