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Rafael Mariano de Bitencourt

Universidade do Sul de Santa Catarina

4 papers in the library · 43 citations · publishing 2020-2026

Papers

Antidepressant and anxiolytic-like effects of ayahuasca in rats subjected to LPS-induced neuroinflammation

Behavioural Brain Research July 14, 2022 Marina Goulart Da Silva, Guilherme Cabreira Daros, Fabiana Pereira Santos et al. 22 citations

Ayahuasca reduced anxiety-like and depressive-like behaviors in rats with neuroinflammation induced by lipopolysaccharide (0.63 mg/kg/mL). Eighty male rats, about 90 days old, were divided into control and LPS groups, with prevention and treatment subgroups. Ayahuasca (4 mL/kg) or saline was given by gavage one hour before or 24 hours after LPS or saline injections. Open field and forced swimming tests measured behavior. LPS rats given ayahuasca showed less anxiety-like behavior in both subgroups. Depressive-like behavior decreased in LPS rats given ayahuasca, in both prevention and treatment subgroups, compared to controls. The findings suggest anxiolytic and antidepressant potential of ayahuasca in neuroinflammation, possibly via antineuroinflammatory effects.

Anti-inflammatory activity of ayahuasca: therapeutical implications in neurological and psychiatric diseases

Behavioural Brain Research November 6, 2020 Marina Goulart Da Silva, Guilherme Cabreira Daros, Rafael Mariano de Bitencourt 21 citations

Ayahuasca, a psychoactive decoction used for millennia by indigenous groups and Amazonian populations, shows therapeutic effects on behavioral disorders by inhibiting monoamine oxidase and activating serotonin receptors. Its pharmacological response also involves anti-inflammatory action, primarily through dimethyltryptamines (N,N-dimethyltryptamine and 5-methoxy-N,N-dimethyltryptamine), which regulate inflammation and immune homeostasis via sigma-1 receptors. Because neuroinflammation underlies many neurological and psychiatric diseases, the available evidence suggests ayahuasca is a promising and very safe therapeutic strategy, as extremely high doses are required for toxicity. However, additional studies are needed to confirm this evidence and fully elucidate the mechanisms involved.

Single exposure to Ayahuasca reverses chronic stress effects on sociability, anxiety, cortisol, and BDNF in zebrafish

Psychopharmacology April 14, 2026 Guilherme Lodetti, Antonio Inserra, Henrique Redivo et al.

A single exposure to ayahuasca reversed behavioral and biochemical changes caused by 14 days of unpredictable chronic stress in adult zebrafish. Stressed fish showed impaired sociability, anxiety-like behavior, hyperactivity, elevated whole-body cortisol, and reduced whole-brain BDNF. Ayahuasca restored sociability, reduced anxiety-like behavior and hyperactivity, normalized cortisol levels, and increased BDNF. These findings suggest ayahuasca can reverse stress-induced behavioral and neuroendocrine alterations, supporting further clinical studies for chronic stress.

As mudanças psicológicas promovidas pela ayahuasca em participantes iniciantes: um estudo observacional longitudinal

Revista Neurociências October 16, 2024 Vitória Pereira de Menezes, Luis Felipe Batista, Vicente Meneguzzo et al.

Mental disorders are common, but treatments are limited by side effects and low efficacy. Ayahuasca, used for millennia by Indigenous peoples, is being explored as an alternative for anxiety and depression. In an observational longitudinal study of 16 first-time participants in Ayahuasca ceremonies in Brazil, anxiety scores decreased significantly one week and three months after use, and depressive symptoms dropped significantly after one week. The authors suggest the results show promise but note that controlled clinical trials with larger samples and longer follow-up are needed for definitive conclusions.