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Molecular Neurobiology

ISSN 0893-7648

2 papers in the library · 57 citations · publishing 2009-2024

Papers

Esketamine Prevents Postoperative Emotional and Cognitive Dysfunction by Suppressing Microglial M1 Polarization and Regulating the BDNF-TrkB Pathway in Ageing Rats with Preoperative Sleep Disturbance

Molecular Neurobiology January 15, 2024 Yuxin Wen, Jiawen Xu, Jiahong Shen et al. 57 citations

Sleep disturbance before surgery worsens postoperative depression and cognitive dysfunction by promoting microglial M1 polarization and disrupting BDNF-TrkB signaling in the brain, leading to emotional changes and cognitive impairments. Treatment with esketamine, the S-enantiomer of ketamine, reversed these behavioral abnormalities by inhibiting microglial M1 polarization and the inflammatory response, thereby improving BDNF-TrkB signaling both in living organisms and in cell cultures. Esketamine also restored impaired hippocampal synaptic plasticity caused by sleep disturbance and surgery. These results suggest that preoperative sleep disruption contributes to postoperative brain complications through inflammatory and neurotrophic mechanisms, and esketamine may offer a protective intervention.

Molecular and Cellular Mechanisms of Ecstasy-Induced Neurotoxicity: An Overview

Molecular Neurobiology June 1, 2009 João Paulo Capela, Helena Carmo, Fernando Remião et al.

MDMA (ecstasy) is a widely abused hallucinogenic drug that can damage nerve cells in both animals and humans. In rats and some mouse strains, it destroys serotonin-producing nerve endings and causes broader brain damage in areas like the cortex, hippocampus, and striatum. In human users, reduced serotonin markers correlate with lasting memory and learning problems. The neurotoxicity involves multiple factors: hyperthermia, metabolism by monoamine oxidase, dopamine oxidation, serotonin transporter activity, nitric oxide and peroxynitrite formation, glutamate excitotoxicity, serotonin 2A receptor activation, and toxic metabolites. This review summarizes the history, pharmacology, metabolism, and cellular/molecular mechanisms of MDMA neurotoxicity to aid development of treatments for long-term psychiatric complications.